Warfarin + Imatinib Mesylate Interaction
Contraindicatedinteraction on record
Description
Warfarin should not be used in patients requiring anticoagulation; use low-molecular weight or standard heparin instead due to CYP2C9 and CYP3A4 metabolism.
Mechanism
Warfarin metabolized by CYP2C9 and CYP3A4; imatinib inhibits CYP3A4
Source: NLP:imatinib mesylate