Tovorafenib + Cyp3a Inhibitors (Moderate And Strong) Interaction

Moderateinteraction on record

Description

CYP2C8 inhibitors are predicted to increase tovorafenib exposure, which may increase the risk of adverse reactions. Avoid coadministration.

Mechanism

Tovorafenib is a CYP2C8 substrate; inhibitors increase its exposure

Source: NLP:tovorafenib