Tolterodine Tartrate + Fluoxetine Interaction

Moderateinteraction on record

Description

Potent CYP2D6 inhibitor that significantly inhibits tolterodine metabolism, resulting in 4.8-fold increase in tolterodine AUC in extensive metabolizers. No dose adjustment required.

Mechanism

CYP2D6 inhibition

Source: NLP:tolterodine tartrate