Teriflunomide + Methotrexate Interaction

Moderateinteraction on record

Description

Teriflunomide may increase exposure of methotrexate via OAT3 and OATP inhibition. Monitor patients and adjust dose as required.

Mechanism

OAT3 and OATP1B1/B3 inhibition

Source: NLP:teriflunomide