Teriflunomide + Methotrexate Interaction
Moderateinteraction on record
Description
Teriflunomide may increase exposure of methotrexate via OAT3 and OATP inhibition. Monitor patients and adjust dose as required.
Mechanism
OAT3 and OATP1B1/B3 inhibition
Source: NLP:teriflunomide