Temsirolimus + Rifampin Interaction
Moderateinteraction on record
Description
Potent CYP3A4/5 inducer decreases sirolimus (primary metabolite) Cmax by 65% and AUC by 56%. Dose adjustment of temsirolimus recommended if alternative cannot be used.
Mechanism
CYP3A4/5 induction
Source: NLP:temsirolimus