Siponimod + Dual Strong Cyp3a4 Moderate Cyp1a2 Inducers Interaction
Majorinteraction on record
Description
Dual moderate CYP2C9/strong CYP3A4 inducers decrease siponimod exposure; concomitant use is not recommended.
Mechanism
CYP2C9/CYP3A4 induction decreases drug exposure
Source: NLP:siponimod