Sensitive Cyp3a Substrates + Nitisinone Interaction
Majorinteraction on record
Description
Nitisinone is a moderate CYP2C9 inhibitor that may increase exposure of co-administered drugs metabolized by CYP2C9, requiring dosage reduction by half and additional adjustments to maintain therapeutic concentrations.
Mechanism
CYP2C9 inhibition
Source: NLP:nitisinone