Sensitive Cyp3a Substrates + Lenacapavir Sodium Interaction
Moderateinteraction on record
Description
YEZTUGO may increase concentrations of sensitive CYP3A substrates, resulting in increased risk of adverse events. Monitoring or dosing adjustments may be needed.
Mechanism
Moderate CYP3A inhibition by lenacapavir
Source: NLP:lenacapavir sodium