Seladelpar Lysine + Cyclosporine Interaction

Moderateinteraction on record

Description

Cyclosporine (dual/multiple inhibitor of OATP1B1, OATP1B3, BCRP) increases seladelpar exposure. Monitor for adverse effects.

Mechanism

Inhibition of drug transporters OATP1B1, OATP1B3, and BCRP

Source: NLP:seladelpar lysine