Rosuvastatin Calcium + Febuxostat Interaction
Majorinteraction on record
Description
Febuxostat increases rosuvastatin exposure more than 1.9-fold, increasing risk of myopathy and rhabdomyolysis. Do not exceed 20 mg rosuvastatin once daily.
Mechanism
CYP2C9 and transporter inhibition
Source: NLP:rosuvastatin calcium