Revefenacin + Rifampin Interaction

Majorinteraction on record

Description

OATP1B1 and OATP1B3 inhibitor that may increase systemic exposure of revefenacin's active metabolite. Coadministration not recommended.

Mechanism

Inhibition of OATP1B1 and OATP1B3 transporters

Source: NLP:revefenacin