Rapamycin + Mifepristone Interaction
Contraindicatedinteraction on record
Description
Mifepristone increases sirolimus exposure; concomitant use is contraindicated due to narrow therapeutic range.
Mechanism
CYP3A inhibition
Source: NLP:mifepristone
Mifepristone increases sirolimus exposure; concomitant use is contraindicated due to narrow therapeutic range.
CYP3A inhibition
Source: NLP:mifepristone