Posaconazole + Rapamycin Interaction
Contraindicatedinteraction on record
Description
Posaconazole increases sirolimus blood concentrations approximately 9-fold, resulting in sirolimus toxicity.
Mechanism
CYP3A4 inhibition
Source: NLP:posaconazole
Posaconazole increases sirolimus blood concentrations approximately 9-fold, resulting in sirolimus toxicity.
CYP3A4 inhibition
Source: NLP:posaconazole