Paroxetine Hydrochloride Hemihydrate + Pimozide Interaction

Contraindicatedinteraction on record

Description

Paroxetine increases pimozide AUC by 151% and Cmax by 62%, leading to increased QT prolongation risk. Contraindicated due to narrow therapeutic index.

Mechanism

CYP2D6 inhibition by paroxetine

Source: NLP:paroxetine hydrochloride hemihydrate