P Gp Or Bcrp Substrates + Vanzacaftor Tezacaftor And Deutivacaftor Interaction

Moderateinteraction on record

Description

Monitor more frequently for adverse reactions. Tezacaftor and deutivacaftor are P-gp inhibitors that increase exposure of P-gp substrates.

Mechanism

P-glycoprotein inhibition increases substrate exposure

Source: NLP:vanzacaftor, tezacaftor, and deutivacaftor