Oxycodone Hydrochloride + Macrolide Antibiotics Eg Erythromycin Interaction

Majorinteraction on record

Description

CYP3A4 inhibitors increase plasma concentration of oxycodone, resulting in increased or prolonged opioid effects, respiratory depression, and sedation.

Mechanism

CYP3A4 inhibition

Source: NLP:oxycodone hydrochloride