Oral Contraceptives + Repotrectinib Interaction
Majorinteraction on record
Description
Repotrectinib decreases progestin or estrogen exposure, reducing contraceptive effectiveness. Avoid concomitant use; use nonhormonal contraception instead.
Mechanism
CYP3A4 induction decreases progestin or estrogen exposure
Source: NLP:repotrectinib