Oral Contraceptives + Omaveloxolone Interaction

Majorinteraction on record

Description

Omaveloxolone weakly induces CYP3A4, which may reduce the efficacy of hormonal contraceptives. Avoid concomitant use with combined hormonal contraceptives, implants, and progestin-only pills.

Mechanism

Weak CYP3A4 induction reduces hormonal contraceptive exposure

Source: NLP:omaveloxolone