Omaveloxolone + Mao Inhibitors Interaction

Majorinteraction on record

Description

Concomitant use results in clinically significant increased exposure of omaveloxolone, which may increase the risk of adverse reactions. Avoid concomitant use; if unavoidable, dosage reduction with monitoring is recommended.

Mechanism

CYP3A4 inhibition increases omaveloxolone exposure

Source: NLP:omaveloxolone