Nicardipine Hydrochloride + Tacrolimus Interaction
Majorinteraction on record
Description
Nicardipine may elevate plasma tacrolimus levels through inhibition of hepatic microsomal enzymes including CYP3A4. Plasma concentrations should be closely monitored and dose adjusted accordingly.
Mechanism
Inhibition of hepatic microsomal enzymes, including CYP3A4
Source: NLP:nicardipine hydrochloride