Nicardipine Hydrochloride + Cyclosporine Interaction

Majorinteraction on record

Description

Nicardipine elevates plasma cyclosporine levels through inhibition of hepatic microsomal enzymes including CYP3A4. Cyclosporine plasma concentrations should be closely monitored and dosage reduced accordingly.

Mechanism

Inhibition of hepatic microsomal enzymes, including CYP3A4

Source: NLP:nicardipine hydrochloride