Neratinib + Strong Or Moderate Cyp3a Inducers Interaction
Contraindicatedinteraction on record
Description
Concomitant use reduces neratinib Cmax and AUC, reducing NERLYNX activity. Avoid concomitant use.
Mechanism
Increased CYP3A4-mediated metabolism of neratinib
Source: NLP:neratinib