Neratinib + Strong Cyp3a4 And P Glycoprotein Inducers Interaction
Contraindicatedinteraction on record
Description
Concomitant use may increase neratinib Cmax and AUC, increasing risk of NERLYNX toxicity. Avoid concomitant use.
Mechanism
Inhibition of P-glycoprotein and moderate CYP3A4-mediated metabolism
Source: NLP:neratinib