Nerandomilast + Mao Inhibitors Interaction

Moderateinteraction on record

Description

Strong CYP3A inhibitors increase exposure of nerandomilast, which may increase the risk of JASCAYD adverse reactions. Dosage reduction to 9 mg twice daily is recommended.

Mechanism

Inhibition of CYP3A metabolism increases nerandomilast exposure

Source: NLP:nerandomilast