Macitentan And Tadalafil + Amiodarone Interaction
Contraindicatedinteraction on record
Description
Moderate dual CYP3A4 and CYP2C9 inhibitor increases macitentan exposure. Avoid concomitant use.
Mechanism
CYP3A4 and CYP2C9 inhibition
Source: NLP:macitentan and tadalafil