Macitentan + Rifampin Interaction
Contraindicatedinteraction on record
Description
Strong CYP3A4 inducer significantly reduces macitentan exposure. Avoid co-administration.
Mechanism
CYP3A4 induction
Source: NLP:macitentan
Strong CYP3A4 inducer significantly reduces macitentan exposure. Avoid co-administration.
CYP3A4 induction
Source: NLP:macitentan