Lofexidine Hydrochloride + Paroxetine Interaction
Moderateinteraction on record
Description
CYP2D6 inhibitor paroxetine increases lofexidine plasma levels by 28%. Monitor for orthostatic hypotension and bradycardia.
Mechanism
CYP2D6 inhibition increases lofexidine absorption
Source: NLP:lofexidine hydrochloride