Linagliptin And Metformin Hydrochloride + Rifampin Interaction
Majorinteraction on record
Description
Strong P-gp or CYP3A4 inducer that decreases linagliptin exposure and may reduce linagliptin efficacy. Alternative treatments are strongly recommended.
Mechanism
Strong P-glycoprotein and CYP3A4 enzyme inducer
Source: NLP:linagliptin and metformin hydrochloride