Ivabradine + Diltiazem Hydrochloride Interaction

Contraindicatedinteraction on record

Description

Concurrent use increases ivabradine exposure and may exacerbate bradycardia and conduction disturbances. Avoid concomitant use.

Mechanism

CYP450 3A4 inhibition by diltiazem increases ivabradine exposure

Source: NLP:diltiazem hydrochloride