Isavuconazonium Sulfate + Lopinavir And Ritonavir Interaction

Moderateinteraction on record

Description

96% increase in isavuconazole exposure when coadministered. Also causes decreased exposure of lopinavir and ritonavir with potential loss of antiviral efficacy.

Mechanism

CYP3A4 inhibition

Source: NLP:isavuconazonium sulfate