Guanfacine + Rifampin Interaction

Majorinteraction on record

Description

CYP3A4 inducer that significantly decreases guanfacine plasma concentrations and exposure. Guanfacine dose increase up to double the target dosage may be needed.

Mechanism

Induction of CYP3A4-mediated metabolism of guanfacine

Source: NLP:guanfacine