Grapefruit Products + Vanzacaftor Tezacaftor And Deutivacaftor Interaction
Moderateinteraction on record
Description
Food or drink containing grapefruit should be avoided. Grapefruit moderately inhibits CYP3A, which may increase exposure of vanzacaftor, tezacaftor, and deutivacaftor.
Mechanism
CYP3A inhibition increases substrate exposure
Source: NLP:vanzacaftor, tezacaftor, and deutivacaftor