Grapefruit Juice + Pexidartinib Hydrochloride Interaction
Moderateinteraction on record
Description
Moderate or strong CYP3A inhibitor that may increase pexidartinib concentrations, increasing incidence and severity of adverse reactions. Reduce TURALIO dosage if concomitant use cannot be avoided.
Mechanism
CYP3A inhibition
Source: NLP:pexidartinib hydrochloride