Grapefruit Juice + Butalbital%2C Acetaminophen%2C Caffeine And Codeine Phosphate Interaction

Majorinteraction on record

Description

CYP3A4 inhibitor may increase codeine plasma concentrations and morphine levels, potentially causing fatal respiratory depression, particularly when added after stable dosing.

Mechanism

Inhibition of CYP3A4, increasing codeine metabolism to morphine via CYP2D6

Source: NLP:butalbital, acetaminophen, caffeine and codeine phosphate