Gemfibrozil + Pioglitazone And Glimepiride Interaction
Majorinteraction on record
Description
Strong CYP2C8 inhibitor significantly increases pioglitazone exposure and half-life. Maximum pioglitazone dose must be limited to 15 mg daily.
Mechanism
CYP2C8 inhibition increases pioglitazone AUC and half-life
Source: NLP:pioglitazone and glimepiride