Famotidine + Tizanidine Interaction

Contraindicatedinteraction on record

Description

Famotidine is a weak CYP1A2 inhibitor and may substantially increase tizanidine blood concentrations, resulting in hypotension, bradycardia, or excessive drowsiness. Avoid concomitant use if possible.

Mechanism

CYP1A2 inhibition

Source: NLP:famotidine