Erlotinib Hydrochloride + Rifampin Interaction

Majorinteraction on record

Description

CYP3A4 and moderate CYP1A2 inducer decreases erlotinib exposure. Increase erlotinib dosage if co-administration is unavoidable.

Mechanism

CYP3A4 and CYP1A2 induction decreases erlotinib plasma concentrations

Source: NLP:erlotinib hydrochloride