Enasidenib Mesylate + Anti Fungal Agents That Are Cyp3a4 Substrates Interaction

Majorinteraction on record

Description

Do not administer enasidenib with anti-fungal agents that are CYP3A substrates due to expected loss of antifungal efficacy.

Mechanism

CYP3A induction leading to decreased antifungal exposure

Source: NLP:enasidenib mesylate