Elagolix And Estradiol And Norethisterone + Mao Inhibitors Interaction

Contraindicatedinteraction on record

Description

OATP1B1 inhibitors that significantly increase elagolix plasma concentrations are contraindicated due to increased risk of elagolix-associated adverse reactions.

Mechanism

OATP1B1 inhibition

Source: NLP:elagolix and estradiol and norethisterone