Dolutegravir Sodium + Etravirine Interaction
Majorinteraction on record
Description
Etravirine significantly reduces plasma concentrations of dolutegravir, reducing therapeutic effect; coadministration with lopinavir/ritonavir, darunavir/ritonavir, or atazanavir/ritonavir may mitigate this effect.
Mechanism
Enzyme induction reducing dolutegravir exposure
Source: NLP:dolutegravir sodium