Darunavir Cobicistat Emtricitabine And Tenofovir Alafenamide + P Gp Or Bcrp Substrates Interaction

Moderateinteraction on record

Description

Co-administration may result in increased plasma concentrations of P-gp substrates due to transporter inhibition.

Mechanism

Cobicistat inhibits P-glycoprotein transporter

Source: NLP:darunavir, cobicistat, emtricitabine, and tenofovir alafenamide