Cyp3a Inhibitors Moderate And Strong + Tovorafenib Interaction

Moderateinteraction on record

Description

CYP2C8 inhibitors are predicted to increase tovorafenib exposure, which may increase the risk of adverse reactions. Avoid coadministration.

Mechanism

Tovorafenib is a CYP2C8 substrate; inhibitors increase its exposure

Source: NLP:tovorafenib