Cyp3a Inducers + Paltusotine Interaction

Moderateinteraction on record

Description

Concomitant use may decrease paltusotine exposure and affect therapeutic response. May require PALSONIFY dosage increase up to three-fold or 120 mg daily, whichever is less.

Mechanism

CYP3A4 induction decreases paltusotine exposure

Source: NLP:paltusotine