Cyp3a Inducers + Olutasidenib Interaction
Majorinteraction on record
Description
Strong CYP3A inducers decrease olutasidenib Cmax and AUC, which may reduce REZLIDHIA efficacy. Avoid concomitant use.
Mechanism
Olutasidenib is a CYP3A substrate; inducers decrease its plasma concentrations
Source: NLP:olutasidenib