Cyp3a Inducers + Elvitegravir Cobicistat Emtricitabine And Tenofovir Alafenam Interaction

Majorinteraction on record

Description

CYP3A inducers increase clearance of elvitegravir and cobicistat, resulting in decreased plasma concentrations and potential loss of therapeutic effect or resistance.

Mechanism

Induction of CYP3A metabolism

Source: NLP:elvitegravir, cobicistat, emtricitabine, and tenofovir alafenamide