Cyp3a Inducers + Dolutegravir Sodium And Rilpivirine Hydrochloride Interaction
Majorinteraction on record
Description
CYP3A4 inducers may decrease rilpivirine plasma concentrations, resulting in loss of virologic response and possible resistance to rilpivirine or NNRTIs.
Mechanism
Induction of cytochrome P450 3A4 metabolism of rilpivirine
Source: NLP:dolutegravir sodium and rilpivirine hydrochloride