Cyclosporine + Atorvastatin Calcium Interaction

Contraindicatedinteraction on record

Description

Significantly increases atorvastatin plasma levels and increases risk of myopathy and rhabdomyolysis. Concomitant use is not recommended.

Mechanism

Inhibition of CYP3A4 and OATP1B1

Source: NLP:atorvastatin calcium