Colchicine + Cyclosporine Interaction

Contraindicatedinteraction on record

Description

Toxicity reported. Dual inhibitor of P-glycoprotein and CYP3A4 causing life-threatening or fatal colchicine toxicity, especially in patients with renal or hepatic impairment.

Mechanism

Inhibition of P-glycoprotein and CYP3A4

Source: NLP:colchicine