Clopidogrel Bisulfate + Repaglinide Interaction

Contraindicatedinteraction on record

Description

Clopidogrel increases repaglinide exposure 3.9-5.1 fold. Avoid concomitant use or adjust dose and monitor closely.

Mechanism

CYP2C8 inhibition by clopidogrel acyl-β-glucuronide metabolite

Source: NLP:clopidogrel bisulfate