Clopidogrel + Repaglinide Interaction

Contraindicatedinteraction on record

Description

Clopidogrel increases repaglinide exposure by 3.9- to 5.1-fold. Avoid concomitant use.

Mechanism

CYP2C8 inhibition by clopidogrel's acyl-β-glucuronide metabolite

Source: NLP:clopidogrel